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Niacin induces PPARγ expression and transcriptional activation in macrophages via HM74 and HM74a-mediated induction of prostaglandin synthesis pathways

Abstract:

HM74 and HM74a have been identified as receptors for niacin. HM74a mediates the pharmacological anti-lipolytic effects of niacin in adipocytes by reducing intracellular cyclic AMP (cAMP) and inhibiting release of free fatty acids into the circulation. In macrophages, niacin induces peroxisome proliferator-activated receptor γ (PPARγ)-dependent and cAMP-dependent expression of genes mediating reverse cholesterol transport, although via an unidentified receptor. We describe constitutive express...

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Publication status:
Published
Peer review status:
Peer reviewed

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Publisher copy:
10.1016/j.bcp.2005.11.019

Authors


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Institution:
University of Oxford
Division:
MSD
Department:
RDM
Sub department:
Weatherall Insti. of Molecular Medicine
Research group:
Cancer Research UK Molecular Oncology Laboratory
Role:
Author
More by this author
Institution:
Institute of Cancer, Sutton, UK
Department:
Cancer Research UK Centre for Cancer Therapeutics
Role:
Author
More by this author
Institution:
Institute of Cancer, Sutton, UK
Department:
Cancer Research UK Centre for Cancer Therapeutics
Role:
Author
More by this author
Institution:
University of Oxford
Division:
MSD
Department:
RDM
Sub department:
Weatherall Insti. of Molecular Medicine
Research group:
Cancer Research UK Molecular Oncology Laboratory
Role:
Author
Cancer Research UK More from this funder
Publisher:
Elsevier Publisher's website
Journal:
Biochemical Pharmacology Journal website
Volume:
71
Issue:
5
Pages:
646-656
Publication date:
2006-02-01
DOI:
ISSN:
0006-2952
Language:
English
Subjects:
UUID:
uuid:a8a5ce26-1079-4f70-878a-ee1cc2aa6ca5
Local pid:
ora:6313
Deposit date:
2012-06-27

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